Universitätsstiftung Hans Vielberth
6th Summer School Medicinal Chemistry at the University of Regensburg
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Program of the conference:

Wednesday, Sept 26, 2012
13.00 h Welcome Armin Buschauer
Thomas Strothotte, Rector of the University of Regensburg
13.10-14.10 h Structural insights into Adenylyl Cyclase inhibitors Stephen R. Sprang
University of Montana, Missoula, MO, USA
14.10-15.10 h Structural insights into opioid receptor function Sébastien Granier
Stanford University, Stanford, CA, USA
15.10-15.40 h

Coffee break


15.40-16.40 h Multiple allosteric sites on muscarinic and FFA1 receptors Nigel Birdsall
National Institute for Medical Research, London, UK
16.40-17.40 h Allosteric modulation of GPCRs: Chemokine receptor CXCR3 as an example Nuška Tschammer
Department of Chemistry and Pharmacy, Emil Fischer Center, University of Erlangen-Nürnberg, DE
17.40- 18.00 h
Coffee break
18.00-19.00 h Structure based GPCR ligand design – use of homology models and crystal structures for lead identification and lead optimization Christofer Tautermann
Boehringer Ingelheim, Biberach, DE
19.00-19.30 h Oral poster presentation
19.30 h Poster session / Beer and bretzel

Thursday, Sept 27, 2012
8.30-9.30 h Drug Design – Solved and Unsolved Problems Hugo Kubinyi
University of Heidelberg, Heidelberg, DE
9.30-10.30 h Structure based drug design for epigenetic targets Wolfgang Sippl
Institute of Pharmacy, Martin-Luther-University Halle-Wittenberg, DE
10.30- 11.00
Coffee break
11.00-12.00 h A Journey in Structure-based Drug Discovery: Inhibitors of IGF1R Kinase (Oncology) and 11ß-HSD1 (Diabetes) Kurt Ritter
Sanofi-Aventis, Frankfurt, DE
12.00-12.30 h Oral poster presentation
12.30- 13.45 h
Lunch break
13.45-14.45 h Argyrin F - a new proteasom inhibitor Markus Kalesse
Institute of Organic Chemistry, University of Hannover, DE
14.45-15.45 h Chemical oncology - converging cancer genetics, structural biology and medicinal chemistry Daniel Rauh
Faculty of Chemistry - Chemical Biology, TU Dortmund, DE
15.45-16.00 h Oral poster presentation
16.00- 16.30
Coffee break
16.30-17.30 h Hedgehog signaling inhibitors for cancer therapy Martial Ruat
Institute of Neurobiology A. Fessard, Gif-Yvette, FR
17.30-18.30 h Kinase-Inhibitors at Bayer Oncology  -   Three Chapters of an Exciting Story Franz von Nussbaum
Bayer HealthCare, Berlin, DE
18.30-18.45 h Oral poster presentation
18.45-20.00 h Poster session
20.00 h Barbecue at the University of Regensburg

Friday, Sept 28, 2012
8.30-9.30 h Change or be changed - Reflections of the workshop "Future in Medicinal Chemistry” Daniel Rauh
Faculty of Chemistry - Chemical Biology, TU Dortmund, DE
9.30-10.30 h Monitoring whole cell responses with label-free biosensors: fancy trend or holistic approach to resolve cellular signaling? Evi Kostenis
Institute of Pharmaceutical Biology, Bonn, DE
10.30- 10.45
Coffee break
10.45-11.45 h Eavesdropping on Cell-Based Assays using Wired Culture Dishes Joachim Wegener
Institute of Analytical Chemistry, University of Regensburg, DE
11.45-12.45 h Ion channels and GPCRs: The age of enlightenment Dirk Trauner
Department of Chemistry,
Ludwig-Maximilians-
University Munich, DE
12.45 h Poster prizes
Concluding remarks

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