Universitätsstiftung Hans Vielberth
6th Summer School Medicinal Chemistry at the University of Regensburg
Registration and Fees
Submission of abstracts
How to get to the venue
Visit Regensburg

Program of the conference:

Wednesday, Sept 26, 2012
13.00 h Welcome Armin Buschauer
Thomas Strothotte, Rector of the University of Regensburg
13.10-14.10 h Structural insights into Adenylyl Cyclase inhibitors Stephen R. Sprang
University of Montana, Missoula, MO, USA
14.10-15.10 h Structural insights into opioid receptor function Sébastien Granier
Stanford University, Stanford, CA, USA
15.10-15.40 h

Coffee break

15.40-16.40 h Multiple allosteric sites on muscarinic and FFA1 receptors Nigel Birdsall
National Institute for Medical Research, London, UK
16.40-17.40 h Allosteric modulation of GPCRs: Chemokine receptor CXCR3 as an example Nuška Tschammer
Department of Chemistry and Pharmacy, Emil Fischer Center, University of Erlangen-Nürnberg, DE
17.40- 18.00 h
Coffee break
18.00-19.00 h Structure based GPCR ligand design – use of homology models and crystal structures for lead identification and lead optimization Christofer Tautermann
Boehringer Ingelheim, Biberach, DE
19.00-19.30 h Oral poster presentation
19.30 h Poster session / Beer and bretzel

Thursday, Sept 27, 2012
8.30-9.30 h Drug Design – Solved and Unsolved Problems Hugo Kubinyi
University of Heidelberg, Heidelberg, DE
9.30-10.30 h Structure based drug design for epigenetic targets Wolfgang Sippl
Institute of Pharmacy, Martin-Luther-University Halle-Wittenberg, DE
10.30- 11.00
Coffee break
11.00-12.00 h A Journey in Structure-based Drug Discovery: Inhibitors of IGF1R Kinase (Oncology) and 11ß-HSD1 (Diabetes) Kurt Ritter
Sanofi-Aventis, Frankfurt, DE
12.00-12.30 h Oral poster presentation
12.30- 13.45 h
Lunch break
13.45-14.45 h Argyrin F - a new proteasom inhibitor Markus Kalesse
Institute of Organic Chemistry, University of Hannover, DE
14.45-15.45 h Chemical oncology - converging cancer genetics, structural biology and medicinal chemistry Daniel Rauh
Faculty of Chemistry - Chemical Biology, TU Dortmund, DE
15.45-16.00 h Oral poster presentation
16.00- 16.30
Coffee break
16.30-17.30 h Hedgehog signaling inhibitors for cancer therapy Martial Ruat
Institute of Neurobiology A. Fessard, Gif-Yvette, FR
17.30-18.30 h Kinase-Inhibitors at Bayer Oncology  -   Three Chapters of an Exciting Story Franz von Nussbaum
Bayer HealthCare, Berlin, DE
18.30-18.45 h Oral poster presentation
18.45-20.00 h Poster session
20.00 h Barbecue at the University of Regensburg

Friday, Sept 28, 2012
8.30-9.30 h Change or be changed - Reflections of the workshop "Future in Medicinal Chemistry” Daniel Rauh
Faculty of Chemistry - Chemical Biology, TU Dortmund, DE
9.30-10.30 h Monitoring whole cell responses with label-free biosensors: fancy trend or holistic approach to resolve cellular signaling? Evi Kostenis
Institute of Pharmaceutical Biology, Bonn, DE
10.30- 10.45
Coffee break
10.45-11.45 h Eavesdropping on Cell-Based Assays using Wired Culture Dishes Joachim Wegener
Institute of Analytical Chemistry, University of Regensburg, DE
11.45-12.45 h Ion channels and GPCRs: The age of enlightenment Dirk Trauner
Department of Chemistry,
University Munich, DE
12.45 h Poster prizes
Concluding remarks

frame Summer School Medicinal Chemistry 2012 frame